• Title of article

    Regioselective Carbon–Carbon Bond Formation in the Effector Domain of Ascomycin

  • Author/Authors

    Amarylla Horvath، نويسنده , , Maximilian A Grassberger، نويسنده , , Gerhard Schulz، نويسنده , , Ewald Haidl، نويسنده , , Hildegard Sperner، نويسنده , , Andrea Steck، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2000
  • Pages
    8
  • From page
    7469
  • To page
    7476
  • Abstract
    Starting from 33-O-silyl-protected ascomycin or its 23,24-dehydration product, regio- and stereo-selective formal aldol reactions under carbon–carbon bond formation at C-22, C-23, or C-24 are demonstrated. Additionally, with the 22-silyl enol ether ascomycin derivative a rhodium(I)-catalysed shift of the 19,20 double bond into the 19,38 exocyclic position is observed at elevated temperature.
  • Keywords
    Aldol reaction , enol ether , ketene acetals , Regiospecificity , Macrocycles
  • Journal title
    Tetrahedron
  • Serial Year
    2000
  • Journal title
    Tetrahedron
  • Record number

    1081253