Title of article :
Synthesis of 5-(sulfamoylmethyl)indoles
Author/Authors :
Joan Bosch، نويسنده , , Tomàs Roca، نويسنده , , Montserrat Armengol، نويسنده , , Dolors Fern?ndez-Forner، نويسنده ,
Issue Information :
هفته نامه با شماره پیاپی سال 2001
Abstract :
The synthesis of 5-(sulfamoylmethyl)indoles bearing a two-carbon chain at C-3 (aminoethyl, acetate, hydroxyethyl, ethyl) either by the Grandberg modification of the Fischer indolization or by intramolecular Heck reaction of suitable o-halotrifluoroacetanilides is reported.
Keywords :
Indoles , indolization , Heck reactions , Metabolites , Drugs
Journal title :
Tetrahedron
Journal title :
Tetrahedron