• Title of article

    Sequential oxopyridinium betaine cycloaddition–palladium catalysed cyclisation–anion capture processes

  • Author/Authors

    Mark R Fielding، نويسنده , , Ronald Grigg، نويسنده , , Visuvanathar Sridharan، نويسنده , , Mark Thornton-Pett، نويسنده , , Christopher J Urch، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2001
  • Pages
    12
  • From page
    7737
  • To page
    7748
  • Abstract
    Katritzkyʹs oxopyridinium betaine cycloaddition is employed to generate bridged bicyclic substrates suitable for our palladium(0) catalysed cyclisation–anion capture methodology. A variety of polycyclic heterocycles have been synthesised via monocyclisation–organotin(IV) capture with or without incorporation of carbon monoxide. Sequential cycloaddition–cyclisation can be performed as a one pot process to deliver substantial gain in molecular complexity.
  • Keywords
    Palladium catalysis , Cyclisation , 1 , 3-dipolar cycloaddition , molecular queuing
  • Journal title
    Tetrahedron
  • Serial Year
    2001
  • Journal title
    Tetrahedron
  • Record number

    1082388