• Title of article

    Double thioalkylation/arylation of nitroarenes with the reduction of nitro- to amino group

  • Author/Authors

    Zbigniew Wr?bel، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2003
  • Pages
    10
  • From page
    101
  • To page
    110
  • Abstract
    Some active bicyclic nitroarenes readily react with an excess of alkyl/arylthiols in the presence of DBU and bis-trimethylsilylacetamide (BSA) in DMF solution, to give dithioalkyl/aryl substituted anilines in moderate to good yields via displacement of ortho- and para-hydrogen atoms with simultaneous reduction of the nitro- to amino-group.
  • Keywords
    Amines , Reduction , bicyclic aromatic compounds , Thiols , Substitution
  • Journal title
    Tetrahedron
  • Serial Year
    2003
  • Journal title
    Tetrahedron
  • Record number

    1083782