• Title of article

    One-pot chemoenzymatic synthesis of protected cyanohydrins

  • Author/Authors

    Thomas Purkarthofer، نويسنده , , Wolfgang Skranc، نويسنده , , Hansj?rg Weber، نويسنده , , Herfried Griengl، نويسنده , , Marcel Wubbolts، نويسنده , , Gerald Scholz، نويسنده , , Peter P?chlauer، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2004
  • Pages
    5
  • From page
    735
  • To page
    739
  • Abstract
    In a chemoenzymatic one-pot reaction of ethyl cyanoformate with benzaldehyde catalyzed by the hydroxynitrile lyase from Prunus amygdalus ethoxycarbonylated (R)-mandelonitrile is formed in a highly enatioselective manner. The reaction was performed both in aqueous and organic media. 1H NMR investigations revealed a two-step procedure consisting of an enzyme-catalyzed addition of HCN, generated by hydrolysis of ethyl cyanoformate, to the aldehyde followed by ethoxycarbonylation of the free cyanohydrin in a second step
  • Keywords
    Cyanohydrins , hydroxynitrile lyase (PaHNL) , Chemoenzymatic synthesis , ethyl cyanoformate
  • Journal title
    Tetrahedron
  • Serial Year
    2004
  • Journal title
    Tetrahedron
  • Record number

    1084740