• Title of article

    Efficient solution phase parallel synthesis of norstatine analogs

  • Author/Authors

    Michael V. Voronkov، نويسنده , , Alexander V. Gontcharov، نويسنده , , Zhi-Min Wang، نويسنده , , Paul F. Richardson، نويسنده , , Hartmuth C. Kolb، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2004
  • Pages
    6
  • From page
    9043
  • To page
    9048
  • Abstract
    The reaction of glycidic amides with various functionalized nitriles to afford norstatine analogs in a regio- and diastereoselective fashion (43–99% yield) is described. Utilizing this chemistry, a 20 membered solution phase library was prepared in two steps featuring three points of diversity.
  • Keywords
    Epoxide , Norstatine , nitrile , solution phase combinatorial chemistry
  • Journal title
    Tetrahedron
  • Serial Year
    2004
  • Journal title
    Tetrahedron
  • Record number

    1087115