• Title of article

    Preparation of 5-diaminomethylenebarbiturates by barbituric acid addition to carbodiimides

  • Author/Authors

    Branko S. Jursic، نويسنده , , Fred Douelle، نويسنده , , Edwin D. Stevens، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2003
  • Pages
    6
  • From page
    3427
  • To page
    3432
  • Abstract
    Through NMR spectroscopic monitoring of barbituric acid addition to carbodiimide, a general synthetic procedure for the preparation of 5-diaminomethylenebarbiturates (DABA) was developed. This procedure is very simple and applicable to the preparation of large quantities of DABA derivatives. Through an X-ray structural study of one of the DABA derivatives, it was established that these compounds have an ylide-type structure with strong charge separation within the molecule.
  • Keywords
    barbituric acid , 5-diaminomethylenebarbiturates , immuno-modulating agents
  • Journal title
    Tetrahedron
  • Serial Year
    2003
  • Journal title
    Tetrahedron
  • Record number

    1087757