Title of article
Efficient synthesis of halohydroxypyridines by hydroxydeboronation
Author/Authors
Anne Sophie Voisin، نويسنده , , Alexandre Bouillon، نويسنده , , Jean-Charles Lancelot، نويسنده , , Sylvain Rault، نويسنده ,
Issue Information
هفته نامه با شماره پیاپی سال 2005
Pages
5
From page
1417
To page
1421
Abstract
This paper describes a general method for the synthesis of halohydroxypyridines from novel halopyridinylboronic acids and esters recently described by some of us. Halopyridinylboronic acids and esters have been efficiently hydroxydeboronated under mild conditions by employing hydrogen peroxide or meta-chloroperbenzoic acid. These hydroxylations take place regioselectively without other oxidation (N-oxide formation).
Keywords
Pyridine , Boronic acids , Hydroxydeboronation
Journal title
Tetrahedron
Serial Year
2005
Journal title
Tetrahedron
Record number
1088365
Link To Document