• Title of article

    Ferric chloride/tetraethyl orthosilicate as an efficient system for synthesis of dihydropyrimidinones by Biginelli reaction

  • Author/Authors

    Ivica Cepanec، نويسنده , , Mladen Litvi?، نويسنده , , Anamarija Bartolin?i?، نويسنده , , Marija Lovri?، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2005
  • Pages
    6
  • From page
    4275
  • To page
    4280
  • Abstract
    An efficient method for the Biginelli reaction of aldehydes, acetoacetate esters and urea employing tetraethyl orthosilicate in the presence of ferric chloride is described. These improved reaction conditions allow the preparation of a wide variety of substituted dihydropyrimidinones (including sterically encumbered ones) in high yields and purity under mild reaction conditions.
  • Keywords
    Biginelli reaction , Tetraethyl orthosilicate , Dihydropyrimidinones , Ferric chloride
  • Journal title
    Tetrahedron
  • Serial Year
    2005
  • Journal title
    Tetrahedron
  • Record number

    1088646