• Title of article

    On the reactivity of ascomycin at the binding domain. Part 3: Reactivity of the binding domain towards diazomethane

  • Author/Authors

    Karl Baumann، نويسنده , , Klemens Hoegenauer، نويسنده , , Hermann Knapp، نويسنده , , Markus Bacher، نويسنده , , Andrea Steck، نويسنده , , Trixie Wagner، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2005
  • Pages
    11
  • From page
    4819
  • To page
    4829
  • Abstract
    A thorough product analysis of the reaction of ascomycin with diazomethane has been performed. Apart from the expected oxiranes (epimeric at C9), a whole range of novel derivatives bearing various modifications in the binding domain were obtained. Proposed mechanisms for their formation and stereochemical aspects are discussed.
  • Keywords
    ascomycin , Diazomethane , Methylene insertion , binding domain , X-ray analysis
  • Journal title
    Tetrahedron
  • Serial Year
    2005
  • Journal title
    Tetrahedron
  • Record number

    1088703