• Title of article

    Microwave-assisted synthesis of 4-amino-3,5-dihalopyridines

  • Author/Authors

    Mark Pichowicz، نويسنده , , Simon Crumpler، نويسنده , , B. Edward McDonald and William L. Siegmann، نويسنده , , Julian Blagg، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2010
  • Pages
    6
  • From page
    2398
  • To page
    2403
  • Abstract
    4-Amino-3,5-dihalopyridines have been efficiently prepared via microwave-assisted nucleophilic aromatic substitution of 3,4,5-trihalopyridines using 1–1.1 equiv of primary and secondary amines. The reaction is also applicable to electron rich arylamines.
  • Keywords
    Coupling , nucleophilic aromatic substitution , Pyridines , Amines , Microwave-assisted synthesis
  • Journal title
    Tetrahedron
  • Serial Year
    2010
  • Journal title
    Tetrahedron
  • Record number

    1100677