• Title of article

    New heteroaromatic aminations on 5-aryl-1,2,4-triazines and 1,2,4,5-tetrazines by palladium catalysis

  • Author/Authors

    Laurent Pellegatti، نويسنده , , Emeline Vedrenne، نويسنده , , Jean-Michel Leger، نويسنده , , Christian Jarry، نويسنده , , Sylvain Routier، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2010
  • Pages
    7
  • From page
    4383
  • To page
    4389
  • Abstract
    The efficient and original palladium-catalyzed amination of 5-Aryl-1,2,4-triazines and 1,2,4,5-tetrazines is reported. This Buchwald–Hartwig type reaction leads to the formation of aminated heterocycles via methylsulfur release. The reaction is optimized and a wide range of amines is used to determine the scope and limitations of this methodology.
  • Journal title
    Tetrahedron
  • Serial Year
    2010
  • Journal title
    Tetrahedron
  • Record number

    1100917