Title of article
An easy synthetic approach to 1,2,3-triazole-fused heterocycles
Author/Authors
Vito Fiandanese، نويسنده , , Giuseppe Marchese، نويسنده , , Angela Punzi، نويسنده , , Francesco Iannone، نويسنده , , Giacomo G. Rafaschieri، نويسنده ,
Issue Information
هفته نامه با شماره پیاپی سال 2010
Pages
8
From page
8846
To page
8853
Abstract
A convenient synthesis of 1,2,3-triazole-fused isoindolines and dihydroisoquinolines in good to excellent yield is reported, starting from easily available terminal alkynes and (2-haloaryl)alkylazides. The method is based upon a cycloaddition reaction, via click chemistry, followed by a transition metal-catalyzed functionalization of a C–H bond.
Keywords
Triazole-fused heterocycles , Cycloaddition , Click chemistry , alkynes , Azides
Journal title
Tetrahedron
Serial Year
2010
Journal title
Tetrahedron
Record number
1102648
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