Title of article
Efficient copper-induced coupling between NH-fluoroalkylated sulfoximines and aryl iodides or bromides
Author/Authors
Yohan Macé، نويسنده , , Bruce Pégot، نويسنده , , Régis Guillot، نويسنده , , Chloée Bournaud، نويسنده , , Martial Toffano، نويسنده , , Giang Vo-Thanh، نويسنده , , Emmanuel Magnier، نويسنده ,
Issue Information
هفته نامه با شماره پیاپی سال 2011
Pages
6
From page
7575
To page
7580
Abstract
A high yielding, simple, and flexible copper-based system for N-arylation of fluorinated sulfoximines is reported. Best results were achieved using copper iodide in combination with DMEDA and Cs2CO3 to provide a wide range of N-arylated perfluoroalkylated sulfoximines. These conditions tolerate a great number of substituents on either aromatic cycle, including heteroaromatic rings, for the N-functionalization.
Keywords
Nitrogen , Sulfur , Sulfoximines , fluorinated ligands , copper
Journal title
Tetrahedron
Serial Year
2011
Journal title
Tetrahedron
Record number
1103698
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