• Title of article

    Synthesis of optically active homotryptophan and its oxygen and sulfur analogues

  • Author/Authors

    Koushik Goswami، نويسنده , , Sibasish Paul، نويسنده , , Sandesh T. Bugde، نويسنده , , Surajit Sinha، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2012
  • Pages
    7
  • From page
    280
  • To page
    286
  • Abstract
    d-Homotryptophan and its sulfur analogue have been synthesized by Sonogashira coupling between 3-iodoheteroarenes and ethynyloxazolidine followed by reduction of triple bond and oxidation of alcohol to acid. l-Homotryptophan and its oxygen analogue have been synthesized from silylated internal alkyne using Larock’s heteroannulation as the key reaction. The alkynyloxazolidines were synthesized from l-serine and l-glutamic acid, respectively.
  • Keywords
    Unnatural amino acid , Alkynyloxazolidine , Sonogashira coupling , Larock’s heteroannulation , Homotryptophan
  • Journal title
    Tetrahedron
  • Serial Year
    2012
  • Journal title
    Tetrahedron
  • Record number

    1104041