• Title of article

    Regioselective N9 alkylation of purine rings assisted by β-cyclodextrin

  • Author/Authors

    Qian Zhang، نويسنده , , Gang Cheng، نويسنده , , Yong-Zhen Huang، نويسنده , , Guirong Qu، نويسنده , , Hong-Ying Niu، نويسنده , , Hai-Ming Guo، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2012
  • Pages
    5
  • From page
    7822
  • To page
    7826
  • Abstract
    Under the assistance of β-cyclodextrin, purine was effectively alkylated at N9 together with up to 99% conversion and good to excellent yield using water as the solvent. High regioselectivity-N9/N7 selectivity>99:1 was attributed to the β-cyclodextrin cavity blocked the N7 of purines ring.
  • Keywords
    Purine , Alkylation , Selectivity , ?-Cyclodextrin
  • Journal title
    Tetrahedron
  • Serial Year
    2012
  • Journal title
    Tetrahedron
  • Record number

    1104932