Author/Authors :
Viktor O. Iaroshenko، نويسنده , , Marcelo Vilches-Herrera، نويسنده , , Ashot Gevorgyan، نويسنده , , Satenik Mkrtchyan، نويسنده , , Knar Arakelyan، نويسنده , , Dmytro Ostrovskyi، نويسنده , , Muhammad S.A. Abbasi، نويسنده , , Linda Supe، نويسنده , , Ani Hakobyan، نويسنده , , Alexander Villinger، نويسنده , , Dmitriy M. Volochnyuk، نويسنده , , Andrei Tolmachev، نويسنده ,
Abstract :
The synthesis of 1-deazapurines and isosteres bearing the exocyclic nitrogen atom at position-1 was developed basing on the formal [3+3]-cyclization reaction of nitro-malonaldehyde with the set of electron-excessive aminoheterocycles. Through the functionalization of the purine-like scaffolds synthesized the diversity of compounds furnished in the possition-1 with aryl, alkinyl, and vinyl rests, were obtained.
Keywords :
heterocyclisation , Electron-excessive aminoheterocycles , Nitro-malonaldehyde , Purine isosteres , fused pyridines
