• Title of article

    A Regioselective Route to 5- and 6-Azaindoles

  • Author/Authors

    Lomberget، Thierry نويسنده , , Radix، Sylvie نويسنده , , Barret، Roland نويسنده ,

  • Issue Information
    روزنامه با شماره پیاپی سال 2005
  • Pages
    -207
  • From page
    208
  • To page
    0
  • Abstract
    The synthesis of 4,7-dimethoxy 5- and 6-azaindoles, a structural unit that is present in recently developed anti-HIV-1 agents, was achieved in a regioselective manner. The developed strategy is based on the appropriate choice of a protecting group during a lithium-mediated formylation step, followed by thermal cyclization of azidoacrylates.
  • Keywords
    pyridines , Metalations , 5- and 6-azaindoles , Azides , regioselectivity
  • Journal title
    Synlett
  • Serial Year
    2005
  • Journal title
    Synlett
  • Record number

    110744

    • Link To Document
    https://search.isc.ac/dl/search/defaultta.aspx?DTC=10&DC=110744