• Title of article

    Synthesis of Functionalized Bicyclic Triazoles from Chiral Aziridines

  • Author/Authors

    Kim، Min Sung نويسنده , , Lee، Won Koo نويسنده , , Ha، Hyun-Joon نويسنده , , Yoon، Hyo Jae نويسنده , , Lee، Baeck Kyong نويسنده , , Kwon، Ji Hyun نويسنده , , Kim، Yongeun نويسنده ,

  • Issue Information
    روزنامه با شماره پیاپی سال 2005
  • Pages
    -2186
  • From page
    2187
  • To page
    0
  • Abstract
    Enantiomerically pure 3-substituted-5-amino-4-hydroxy-5,6-dihydro-4H-pyrrolo[1,2-c][1,2,3]triazoles were synthesized efficiently from the sequential reactions including a regioselective ring-opening of 1-aziridine-2-yl-propargylic alcohols by azidotrimethylsilane and the subsequent intramolecular 1,3-dipolar cycloaddition between alkyne and azide.
  • Keywords
    Azide , Cycloaddition , aziridine , Alkyne , triazole
  • Journal title
    Synlett
  • Serial Year
    2005
  • Journal title
    Synlett
  • Record number

    110798