• Title of article

    Reversal of Enantioselectivity by Catalyst Protonation: Asymmetric ­Hydrocyanation of Imines with Oxazaborolidines

  • Author/Authors

    Berkessel، Albrecht نويسنده , , Mukherjee، Santanu نويسنده , , Lex، Johann نويسنده ,

  • Pages
    -40
  • From page
    41
  • To page
    0
  • Abstract
    A new application of chiral oxazaborolidines in asymmetric transformation, namely the hydrocyanation of imines, is described. The effect of protonation of these catalysts on the reactivity and enantioselectivity of hydrocyanations is studied. Significant increase in reaction rate is observed upon protonation of the catalysts, along with the reversal of the sense of stereoinduction.
  • Keywords
    oxazaborolidine , Asymmetric Catalysis , hydrocyanation , Imine , Protonation
  • Journal title
    Astroparticle Physics
  • Record number

    110880