• Title of article

    Synthesis of 7-cycloalkylimino substituted 3-amino-6-fluoro-2-methyl-3H-quinazolin-4-ones

  • Author/Authors

    Nosova، نويسنده , , Emiliya V. and Lipunova، نويسنده , , Galina N. and Slepukhin، نويسنده , , Pavel A. and Charushin، نويسنده , , Valery N.، نويسنده ,

  • Issue Information
    روزنامه با شماره پیاپی سال 2013
  • Pages
    3
  • From page
    63
  • To page
    65
  • Abstract
    A versatile pathway for the synthesis of 7-cycloalkylimino substituted 3-amino-6-fluoro-2-methyl-3H-quinazolin-4-ones from 4,5-difluoroanthranylic acid has been advanced. Nucleophilic amination–defluorination reaction of the 6,7-difluoro derivative of 3-amino-2-methyl-3H-quinazolin-4-one has been established to occur at position 7, as shown by X-ray crystallographic analysis.
  • Keywords
    Fluorine-containing quinazolinones , 3-Aminoquinazolin-4-ones , Nucleophilic displacement reactions , X-ray crystallography
  • Journal title
    Journal of Fluorine Chemistry
  • Serial Year
    2013
  • Journal title
    Journal of Fluorine Chemistry
  • Record number

    1611937