• Title of article

    Highly efficient Cu(I)-catalyzed trifluoromethylation of aryl(heteroaryl) enol acetates with CF3 radicals derived from CF3SO2Na and TBHP at room temperature

  • Author/Authors

    Lu، نويسنده , , Yang and Li، نويسنده , , Yaming and Zhang، نويسنده , , Zhuo-Rong and Jin، نويسنده , , Kun and Duan، نويسنده , , Chunying، نويسنده ,

  • Issue Information
    روزنامه با شماره پیاپی سال 2014
  • Pages
    6
  • From page
    128
  • To page
    133
  • Abstract
    An efficient method for the Cu(I)-catalyzed synthesis of α-trifluoromethyl ketones via the addition of CF3 to aryl(heteroaryl) enol acetates by using the readily available CF3SO2Na (Langlois reagent) has been developed. The reaction is experimentally simple and carried out at room temperature, providing good to excellent yields with wide functional group tolerance.
  • Keywords
    trifluoromethylation , Enol acetates , Synthetic methods , radical addition , ?-CF3 ketone
  • Journal title
    Journal of Fluorine Chemistry
  • Serial Year
    2014
  • Journal title
    Journal of Fluorine Chemistry
  • Record number

    1612244