• Title of article

    Regioselective synthesis of various prodrugs of ganciclovir

  • Author/Authors

    Gao، نويسنده , , Hongwu and Mitra، نويسنده , , Ashim K، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2000
  • Pages
    6
  • From page
    1131
  • To page
    1136
  • Abstract
    High-yield regioselective syntheses of 9-[(1,3-dihydroxy-2-propoxy)methyl]guanine mono-, di- and tri-substitution derivatives as potential prodrugs were accomplished via one or multisteps. Two amino acid esters of ganciclovir were synthesized as water-soluble prodrugs, which form protonated cations in pH 7.4 phosphate buffer.
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2000
  • Journal title
    Tetrahedron Letters
  • Record number

    1636434