• Title of article

    Synthesis of aspartimide-free protected peptides on base-labile functionalized resins

  • Author/Authors

    Rabanal، نويسنده , , Francesc and Pastor، نويسنده , , Jose J and Nicolلs، نويسنده , , Ernesto and Albericio، نويسنده , , Fernando and Giralt*، نويسنده , , Ernest، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2000
  • Pages
    4
  • From page
    8093
  • To page
    8096
  • Abstract
    Aspartimide prone sequence containing protected peptides are successfully synthesized in solid phase by using the bifunctional linker N-[(9-hydroxymethyl)-2-fluorenyl] succinamic acid (HMFS) in combination with morpholine as the cleavage reagent. Access to high purity peptide synthons opens a straightforward way to the synthesis of large proteins by convergent strategies.
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2000
  • Journal title
    Tetrahedron Letters
  • Record number

    1639334