Title of article
Synthesis of a [2]benzazepine analogue of clavizepine
Author/Authors
Garc??a، نويسنده , , Alberto and Paz-Estivill، نويسنده , , Sonia and Dom??nguez، نويسنده , , Domingo، نويسنده ,
Issue Information
هفته نامه با شماره پیاپی سال 2001
Pages
3
From page
665
To page
667
Abstract
The synthesis of N-tosylbenzopyran[2]benzazepinone 2 using a simple protocol for assembly of an azepine ring on the xanthene skeleton is described. Formation of the CC bond between C9 of the xanthen-9-ol 7 and the β-C of N-tosyl aminoacetaldehyde dimethyl acetal leads to 10, which upon treatment with formaldehyde undergoes ring closure.
Keywords
xanthenes , acetals , amino aldehydes , benzazepines , polycyclic heterocyclic compounds
Journal title
Tetrahedron Letters
Serial Year
2001
Journal title
Tetrahedron Letters
Record number
1641380
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