• Title of article

    Synthesis of a [2]benzazepine analogue of clavizepine

  • Author/Authors

    Garc??a، نويسنده , , Alberto and Paz-Estivill، نويسنده , , Sonia and Dom??nguez، نويسنده , , Domingo، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2001
  • Pages
    3
  • From page
    665
  • To page
    667
  • Abstract
    The synthesis of N-tosylbenzopyran[2]benzazepinone 2 using a simple protocol for assembly of an azepine ring on the xanthene skeleton is described. Formation of the CC bond between C9 of the xanthen-9-ol 7 and the β-C of N-tosyl aminoacetaldehyde dimethyl acetal leads to 10, which upon treatment with formaldehyde undergoes ring closure.
  • Keywords
    xanthenes , acetals , amino aldehydes , benzazepines , polycyclic heterocyclic compounds
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2001
  • Journal title
    Tetrahedron Letters
  • Record number

    1641380