Title of article :
Direct amination of β-oxo esters
Author/Authors :
Fioravanti، نويسنده , , Stefania and Morreale، نويسنده , , Alberto and Pellacani، نويسنده , , Lucio and Tardella، نويسنده , , Paolo A، نويسنده ,
Issue Information :
هفته نامه با شماره پیاپی سال 2001
Abstract :
The reaction of NsONHCO2Et, in the presence of CaO, with β-oxo esters gives the corresponding aminated products in yields up to 58%. A substrate carrying the Oppolzer sultam undergoes amination with 40% diastereoselectivity.
Keywords :
amination , keto acids and derivatives , amino acids and derivatives , Carbamates
Journal title :
Tetrahedron Letters
Journal title :
Tetrahedron Letters
