• Title of article

    Efficient synthesis of purine analogues: an FeCl3–SiO2-promoted cyclization reaction of 4,5-diaminopyrimidines with aldehydes leading to 6,8,9-trisubstituted purines

  • Author/Authors

    Dang، نويسنده , , Qun and Brown، نويسنده , , Brian S and Erion، نويسنده , , Mark D، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2000
  • Pages
    4
  • From page
    6559
  • To page
    6562
  • Abstract
    6,8,9-Trisubstituted purine analogues were efficiently synthesized via cyclization of 6-chloro-4,5-diaminopyrimidines and various aldehydes promoted by FeCl3–SiO2. Fe(III) chloride on silica gel has a dual role of a dehydration agent and an oxidant, and was conveniently removed during work-up by filtration.
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2000
  • Journal title
    Tetrahedron Letters
  • Record number

    1642824