• Title of article

    Solid-phase synthesis of functionalized tropane derivatives via 1,3-dipolar cycloaddition

  • Author/Authors

    Caix-Haumesser، نويسنده , , Sandrine and Hanna، نويسنده , , Issam and Lallemand، نويسنده , , Jean-Yves and Peyronel، نويسنده , , Jean-François، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2001
  • Pages
    3
  • From page
    3721
  • To page
    3723
  • Abstract
    1,3-Dipolar cycloaddition of 3-oxidopyridinium betaine to activated olefins on solid-phase leads to resin-bound 8-azabicyclo[3.2.1]octenones which undergo further transformations such as 1,4-addition of nucleophiles. Cleavage of benzyl linker is achieved using acid chlorides in the presence of potassium iodide to give substituted tropane derivatives.
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2001
  • Journal title
    Tetrahedron Letters
  • Record number

    1644968