Title of article
α-(Trifluoromethyl)ethenyl boronic acid as a useful trifluoromethyl containing building block. Preparation and palladium-catalysed coupling with aryl halides
Author/Authors
Jiang، نويسنده , , Biao and Wang، نويسنده , , Quan-Fu and Yang، نويسنده , , Cai-Guang and Xu، نويسنده , , Min، نويسنده ,
Issue Information
هفته نامه با شماره پیاپی سال 2001
Pages
3
From page
4083
To page
4085
Abstract
α-(Trifluoromethyl)ethenyl boronic acid was conveniently prepared from the reaction of readily available 2-bromotrifluoropropene with alkyl borate and magnesium in one-pot. This boronic acid can undergo palladium-catalysed coupling reactions with aryl halides to afford a series of useful α-(trifluoromethyl)styrene derivatives in high yield.
Keywords
Suzuki cross-coupling reaction , ?-(trifluoromethyl)ethenyl boronic acid
Journal title
Tetrahedron Letters
Serial Year
2001
Journal title
Tetrahedron Letters
Record number
1645261
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