Title of article
Solid-phase Friedel–Crafts acylation on polystyrene resins-synthesis of antiepiletic 1-aryl-3,5-dihydro-4H-2,3-benzodiazepin-4-ones
Author/Authors
Bevacqua، نويسنده , , Francesca and Basso، نويسنده , , Andrea and Gitto، نويسنده , , Rosaria and Bradley، نويسنده , , Mark and Chimirri، نويسنده , , Alba، نويسنده ,
Issue Information
هفته نامه با شماره پیاپی سال 2001
Pages
3
From page
7683
To page
7685
Abstract
Friedel–Crafts acylation with various acyl chlorides of resin-bound 3,4-dimethoxyphenylacetate afforded resin bound ketones which, following treatment with hydrazine, were converted into the corresponding 2,3-benzodiazepines in good yields and purities.
Keywords
Friedel–Crafts acylation , solid-phase synthesis , 2 , 3-benzodiazepines
Journal title
Tetrahedron Letters
Serial Year
2001
Journal title
Tetrahedron Letters
Record number
1647918
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