• Title of article

    O-(7-Azabenzotriazol-1-yl)-1,1,3,3-tetramethyluronium hexafluorophosphate–1-hydroxy-7-azabenzotriazole–copper(II) chloride: a promising epimerization-free segment coupling system for peptide synthesis

  • Author/Authors

    Nishiyama، نويسنده , , Yasuhiro and Ishizuka، نويسنده , , Sou and Kurita، نويسنده , , Keisuke، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2001
  • Pages
    3
  • From page
    8789
  • To page
    8791
  • Abstract
    Simultaneous use of 1-hydroxy-7-azabenzotriazole and CuCl2 with O-(7-azabenzotriazol-1-yl)-1,1,3,3-tetramethyluronium hexafluorophosphate has been found to eliminate the enantiomerization of the carboxy-terminal amino acid residue in peptide synthesis by the segment condensation strategy.
  • Keywords
    1 , peptide synthesis , 3-tetramethyluronium hexafluorophosphate , Copper(II) chloride , epimerization suppressant , 1-hydroxy-7-azabenzotriazole , O-(7-azabenzotriazol-1-yl)-1 , 3
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2001
  • Journal title
    Tetrahedron Letters
  • Record number

    1648597