Title of article
Polymer-assisted solution-phase parallel synthesis of dipeptide p-nitroanilides and dipeptide diphenyl phosphonates
Author/Authors
Kristel Senten، نويسنده , , Kristel and Van der Veken، نويسنده , , Pieter and Bal، نويسنده , , Gunther and Haemers، نويسنده , , Achiel and Augustyns، نويسنده , , Koen، نويسنده ,
Issue Information
هفته نامه با شماره پیاپی سال 2001
Pages
4
From page
9135
To page
9138
Abstract
This letter describes the parallel synthesis of dipeptide p-nitroanilides (1) and dipeptide diphenyl phosphonates (2), compounds that can be used as substrates and irreversible inhibitors for the rapid profiling of dipeptidyl peptidases. A polymer-assisted solution-phase synthesis was used for a rapid and clean coupling between easily available building blocks.
Keywords
dipeptide p-nitroanilides , amide coupling , dipeptide diphenyl phosphonates , polymer-assisted solution-phase synthesis
Journal title
Tetrahedron Letters
Serial Year
2001
Journal title
Tetrahedron Letters
Record number
1648851
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