• Title of article

    Original and efficient method for the preparation of N-aminoamide pseudodipeptides in high optical purity

  • Author/Authors

    Brosse، نويسنده , , Nicolas and Grandeury، نويسنده , , Arnaud and Jamart-Grégoire، نويسنده , , Brigitte، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2002
  • Pages
    3
  • From page
    2009
  • To page
    2011
  • Abstract
    N-Aminoamide pseudodipeptides ZAAΨ[CO-N(NPht)]-AAOR can be easily obtained via the Mitsunobu protocol by using α-hydroxyesters as alcohol partners and aminoacid phthaloyl hydrazide derivatives as acidic partners. The direct conversion of the phthaloyl group into tert-butyloxycarbonyl can be performed in a three-stage one-pot protocol.
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2002
  • Journal title
    Tetrahedron Letters
  • Record number

    1650494