Title of article
Aza-Diels–Alder/intramolecular Heck cyclization approach to the tetrahydro-β-carboline skeleton of the ajmaline/sarpagine alkaloids
Author/Authors
Kuethe، نويسنده , , Jeffrey T. and Wong، نويسنده , , Audrey and Davies، نويسنده , , Ian W. and Reider، نويسنده , , Paul J.، نويسنده ,
Issue Information
هفته نامه با شماره پیاپی سال 2002
Pages
4
From page
3871
To page
3874
Abstract
The aza-Diels–Alder reactions of 2-iodo-3-indoleacetaldehydes in the presence of zinc triflate provides 2-(2-iodoindolylmethyl)-4-pyridones in high yield. Palladium-mediated intramolecular Heck cyclization gives access to the tetracyclic tetrahydro-β-carboline framework of the ajmaline/sarpagine alkaloids.
Journal title
Tetrahedron Letters
Serial Year
2002
Journal title
Tetrahedron Letters
Record number
1651826
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