• Title of article

    Convenient synthesis of Cbz-protected β-amino ketones by a copper-catalysed conjugate addition reaction

  • Author/Authors

    Wabnitz، نويسنده , , Tobias C and Spencer، نويسنده , , Jonathan B، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2002
  • Pages
    4
  • From page
    3891
  • To page
    3894
  • Abstract
    A convenient synthesis of Cbz-protected β-amino ketones is reported. Benzyl carbamates and α,β-unsaturated ketones furnish the conjugate addition products in the presence of a Cu(II) catalyst under mild conditions. Other weakly basic nitrogen nucleophiles can also be used in this reaction.
  • Keywords
    benzyl carbamate , conjugate addition , Copper , ?-amino ketones , nitrogen nucleophiles
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2002
  • Journal title
    Tetrahedron Letters
  • Record number

    1651839