• Title of article

    A short synthesis of the C15–C21 segment of (+)-discodermolide, based on an asymmetric approach from achiral 2-methyl-1,3-propanediol to versatile enantiopure stereotriads

  • Author/Authors

    Shahid، نويسنده , , Kazi A. and Li، نويسنده , , Yong-Nan and Okazaki، نويسنده , , Momotoshi and Shuto، نويسنده , , Yoshihiro and Goto، نويسنده , , Fumitaka and Kiyooka، نويسنده , , Syun-ichi، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2002
  • Pages
    4
  • From page
    6373
  • To page
    6376
  • Abstract
    A new approach was developed to versatile enantiopure stereotriads using chiral oxazaborolidinone-promoted asymmetric aldol reaction of a racemic aldehyde with a bromo silyl nucleophile. A short synthesis of the C15–C21 segment of (+)-discodermolide was achieved by elongation of one of the stereotriads with further diastereoselective aldol reaction with the same nucleophile.
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2002
  • Journal title
    Tetrahedron Letters
  • Record number

    1653526