Practical acid-catalyzed acylation of sulfonamides with carboxylic acid anhydrides
Author/Authors :
Martin، نويسنده , , Michael T and Roschangar، نويسنده , , Frank and Eaddy، نويسنده , , John F، نويسنده ,
Issue Information :
هفته نامه با شماره پیاپی سال 2003
Pages :
3
From page :
5461
To page :
5463
Abstract :
A highly efficient reaction between sterically and electronically diverse sulfonamides and carboxylic acid anhydrides to furnish monoacylated N-acylsulfonamides is described. This represents the first systematic disclosure of the scope of sulfuric acid-catalyzed acylation of sulfonamides.