• Title of article

    Effect of the alkyl chain length of 1,1′-binaphthyl esters in lipase-catalyzed amidation

  • Author/Authors

    Aoyagi، نويسنده , , Naoto and Kawauchi، نويسنده , , Shinji and Izumi، نويسنده , , Taeko، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2003
  • Pages
    4
  • From page
    5609
  • To page
    5612
  • Abstract
    Lipase-catalyzed amidation of 2-[2-(ethoxycarbonyl)ethyl]-1,1′-binaphthyl [(±)-3] yielded optically active (S)-3 and 2-[2-(2-cyanoethylaminocarbonyl)ethyl]-1,1′-binaphthyl [(R)-6a] with high enantiomeric excess. For these lipase-catalyzed amidations, the optimal alkyl chain length between the binaphthyl ring and the ester group was determined to be an ethylene spacer.
  • Keywords
    Binaphthyl , Suzuki cross-coupling , Lipase , Amidation , Aminolysis
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2003
  • Journal title
    Tetrahedron Letters
  • Record number

    1653607