• Title of article

    Total syntheses of aminomethyl-C-dideoxyglycopyranosides and their quinamides

  • Author/Authors

    Vyacheslav V. and Gremyachinskiy، نويسنده , , Dmitriy E and Samoshin، نويسنده , , Vyacheslav V. and Gross، نويسنده , , Paul H، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2003
  • Pages
    4
  • From page
    6587
  • To page
    6590
  • Abstract
    Lewis acid promoted cyclization of homoallylic alcohol 1 with acetal 2 gave 4-chloro-2-phthalimidomethyl-6-methyltetrahydropyrans. Their dehydrochlorination produced two regioisomeric dihydropyrans. Subsequent cis- and trans-dihydroxylation gave four racemic dihydroxy-6-methyl-2-phthalimidomethyl tetrahydropyrans. They were deprotected and N-acylated with a chiral quinic acid lactone, producing a library of four diastereomeric mixtures of novel C-pseudodisaccharides, which were separable after derivatization.
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2003
  • Journal title
    Tetrahedron Letters
  • Record number

    1654174