Title of article
An efficient route to 4-(substituted benzyl)piperidines
Author/Authors
Furman، نويسنده , , Bart?omiej and Dziedzic، نويسنده , , Magdalena، نويسنده ,
Issue Information
هفته نامه با شماره پیاپی سال 2003
Pages
4
From page
8249
To page
8252
Abstract
A novel approach to 4-(substituted benzyl)piperidines has been developed. The key steps involve the cyclization of imines bearing an allylsilane in the side-chain followed by the palladium-catalyzed cross-coupling of the resulting 4-methylenepiperidine with organoboronic acids under an atmosphere of oxygen.
Keywords
Cyclisation , Heck reaction , piperidines
Journal title
Tetrahedron Letters
Serial Year
2003
Journal title
Tetrahedron Letters
Record number
1655364
Link To Document