Title of article
New synthetic approaches to CNS drugs. A straightforward, efficient synthesis of tetrahydroindol-4-ones and tetrahydroquinolin-5-ones via palladium-catalyzed oxidation of hydroxyenaminones
Author/Authors
Pita، نويسنده , , Beatriz and Masaguer، نويسنده , , Christian F. and Raviٌa، نويسنده , , Enrique، نويسنده ,
Issue Information
هفته نامه با شماره پیاپی سال 2002
Pages
4
From page
7929
To page
7932
Abstract
We have developed a facile and efficient synthesis of new conformationally restricted butyrophenones in the indole and quinoline series via palladium-catalyzed oxidation of hydroxyenaminones, and subsequent cyclization followed by spontaneous aromatization.
Keywords
enamines , tetrahydroindoles , cyclic ketones , tetrahydroquinolines
Journal title
Tetrahedron Letters
Serial Year
2002
Journal title
Tetrahedron Letters
Record number
1658776
Link To Document