• Title of article

    Synthesis of 2,3-diaminodihydropyrroles via thioimidate cyclopropane rearrangement

  • Author/Authors

    Kuduk، نويسنده , , Scott D and Ng، نويسنده , , Christina L. Chang، نويسنده , , Ronald K and Bock، نويسنده , , Mark G، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2003
  • Pages
    4
  • From page
    1437
  • To page
    1440
  • Abstract
    The synthesis of novel 2,3-diaminodihydropyrroles is reported. The key step is a thiomethylimidate cyclopropane rearrangement to afford a pyrrolothiomethylimidate intermediate. Reaction of this intermediate with amines produced the title compounds in good yields. The scope and mechanism of the reaction is discussed.
  • Keywords
    Cyclopropane , Imidate , dihydropyrroles , Rearrangement
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2003
  • Journal title
    Tetrahedron Letters
  • Record number

    1660642