Title of article
The Bohlmann–Rahtz route to functionalised pyridine scaffolds and their use in library synthesis
Author/Authors
Bashford، نويسنده , , Katherine E. and Burton، نويسنده , , Matthew B. and Cameron، نويسنده , , Stuart and Cooper، نويسنده , , Anthony L. and Hogg، نويسنده , , Rebecca D. and Kane، نويسنده , , Peter D. and MacManus، نويسنده , , David A. and Matrunola، نويسنده , , Christopher A. and Moody، نويسنده , , Christopher J. and Robertson، نويسنده , , Avril A.B. and Warne، نويسنده , , Mark R.، نويسنده ,
Issue Information
هفته نامه با شماره پیاپی سال 2003
Pages
3
From page
1627
To page
1629
Abstract
The Bohlmann–Rahtz reaction has been used to prepare 2,3,6-trisubstituted pyridines suitable for use in library synthesis. The synthesis of piperidine substituted nicotinic acid derivative 9 has been optimised and carried out on a large scale to give ca. 500 g of scaffold which was used in the generation of the pyridine library 11.
Journal title
Tetrahedron Letters
Serial Year
2003
Journal title
Tetrahedron Letters
Record number
1660773
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