• Title of article

    Access to novel substituted diazaadamantanes via semi-natural tetrahydrocytisine

  • Author/Authors

    Ivachtchenko، نويسنده , , Alexandre V. and Khvat، نويسنده , , Alexandre and Tkachenko، نويسنده , , Sergey E. and Sandulenko، نويسنده , , Yuri B. and Vvedensky، نويسنده , , Vladimir Y.، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2004
  • Pages
    4
  • From page
    6733
  • To page
    6736
  • Abstract
    Novel 1,3-diazaadamantane structures 3 and 6 were prepared from tetrahydro(−)-cytisine 1 using intermolecular conversions within the bispidine moiety. 2-Oxo derivative 6 was synthesized using a microwave-assisted procedure, which reduces the reaction time and increases the purity of the crude reaction mixture. Alternative possibilities of intermolecular cyclizations were also explored. Though less successful, they provided interesting insights into the chemistry of bispidine systems.
  • Keywords
    Tetrahydro(?)-cytisine , (1S , 1 , 3-Diazaadamantane , Microwave-assisted , Intermolecular cyclizations , 5S)-1 , 7*]decanes
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2004
  • Journal title
    Tetrahedron Letters
  • Record number

    1843139