Title of article :
First example of the C-alkylation of indoles with Baylis–Hillman acetates
Author/Authors :
Yadav، نويسنده , , J.S. and Reddy، نويسنده , , B.V. Subba and Basak، نويسنده , , A.K. and Narsaiah، نويسنده , , A.V. and Prabhakar، نويسنده , , A. and Jagadeesh، نويسنده , , B.، نويسنده ,
Issue Information :
هفته نامه با شماره پیاپی سال 2005
Pages :
3
From page :
639
To page :
641
Abstract :
Baylis–Hillman acetates undergo SN2′ allylic substitution with indoles in the presence of 20 mol % of indium tribromide under mild conditions to afford a new class of substituted indoles in high yields with (E)-stereoselectivity. The stereochemistry of the products was assigned by various NMR experiments.
Keywords :
Indium compounds , allylic substitution , heteroaromatics
Journal title :
Tetrahedron Letters
Serial Year :
2005
Journal title :
Tetrahedron Letters
Record number :
1844564
Link To Document :
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