Title of article
First efficient synthesis of novel oxophenyl-arcyriaflavin analogs
Author/Authors
Bourderioux، نويسنده , , Aurélie and Routier، نويسنده , , Sylvain and Bénéteau، نويسنده , , Valérie and Mérour، نويسنده , , Jean-Yves، نويسنده ,
Issue Information
هفته نامه با شماره پیاپی سال 2005
Pages
4
From page
6071
To page
6074
Abstract
New oxophenylarcyriaflavins were synthesized in a few efficient steps. The key steps involved at first a palladium cross-coupling between the 3-bromo-4-(1H-indol-3-yl)1-methylpyrrole-2,5-dione and the 2-formylphenylboronic acid or a methyl 2-trialkylstannylbenzoate, followed by an intramolecular acylation in a C-2 indolic position. All the sequence was carried out without any indolic protective group.
Keywords
Anticancer agents , Indolocarbazoles synthesis , Arcyriaflavin
Journal title
Tetrahedron Letters
Serial Year
2005
Journal title
Tetrahedron Letters
Record number
1846558
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