Author/Authors :
Hoarau، نويسنده , , Christophe and Du Fou de Kerdaniel، نويسنده , , Alexis and Bracq، نويسنده , , Nicolas and Grandclaudon، نويسنده , , Pierre and Couture، نويسنده , , Axel and Marsais، نويسنده , , Francis، نويسنده ,
Abstract :
The efficient and regioselective palladium-catalyzed C-2 arylation of ethyl 4-oxazolecarboxylate 1 with phenyliodide is described. The different parameters (solvent, base, ligand and catalyst) for the optimal conditions of this arylation process have been screened.
Keywords :
Ethyl 4-oxazolecarboxylate , Direct coupling , PALLADIUM , aryloxazoles
