Title of article :
Epoxide opening with amino acids: improved synthesis of hydroxyethylamine dipeptide isosteres
Author/Authors :
Babi?، نويسنده , , Andrej and Sova، نويسنده , , Matej and Gobec، نويسنده , , Stanislav and Pe?ar، نويسنده , , Slavko، نويسنده ,
Issue Information :
هفته نامه با شماره پیاپی سال 2006
Abstract :
The amino acid opening of epoxides, catalyzed by calcium trifluoromethanesulfonate with short reaction times is described. The method can be used in a straightforward route for the preparation of hydroxyethylamine dipeptide isosteres.
Keywords :
Hydroxyethylamine dipeptide isosteres , Calcium trifluoromethanesulfonate , epoxides , Peptidomimetics , Aminolysis , proteases
Journal title :
Tetrahedron Letters
Journal title :
Tetrahedron Letters