• Title of article

    Practical Cu-catalyzed amination of functionalized heteroaryl halides

  • Author/Authors

    Yeh، نويسنده , , Vince S.C. and Wiedeman، نويسنده , , Paul E.، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2006
  • Pages
    6
  • From page
    6011
  • To page
    6016
  • Abstract
    The amination of a variety of highly functionalized heterocyclic bromides has been accomplished using a CuI/proline catalyst system. The current study significantly expanded the scope of the reaction by using examples relevant to drug discovery programs and has demonstrated reaction rate acceleration using microwave heating.
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2006
  • Journal title
    Tetrahedron Letters
  • Record number

    1852028