Title of article :
Preparation of enantiopure 2-acylazetidines and their reactions with chloroformates
Author/Authors :
Ma، نويسنده , , Sang-Ho and Yoon، نويسنده , , Doo-Ha and Ha، نويسنده , , Hyun Joon and Lee، نويسنده , , Won Koo، نويسنده ,
Issue Information :
هفته نامه با شماره پیاپی سال 2007
Abstract :
Enantiopure 1-phenylethylazetidine-2-carboxylates and 2-acylazetidines were prepared and reacted with chloroformates to yield α-chloro-γ-amino butyric acid esters and ketones from ring opening reaction of azetidinium ion intermediate in a completely regio- and stereoselective manner.
Keywords :
?-Chloro-?-amino butyric acid esters , Azetidine-2-carboxylate , 2-Acylazetidine , Chloroformate , Ring opening
Journal title :
Tetrahedron Letters
Journal title :
Tetrahedron Letters
